Home GPCR & G Protein Sigma Receptor agonist Carbetapentane For research use only.

Carbetapentane

Synonyms: Pentoxyverine, CB

Carbetapentane (Pentoxyverine, CB) is an antitussive anticonvulsant nonselective sigma-1 (σ1) agonist.

Carbetapentane Chemical Structure

Carbetapentane Chemical Structure

CAS No. 77-23-6

Purity & Quality Control

Carbetapentane Related Products

Biological Activity

Description Carbetapentane (Pentoxyverine, CB) is an antitussive anticonvulsant nonselective sigma-1 (σ1) agonist.
Targets
σ1 [1]
NCT Number Recruitment Conditions Sponsor/Collaborators Start Date Phases
NCT05312372 Withdrawn
Esophageal Squamous Cell Carcinoma
Institut de Recherches Internationales Servier|ADIR a Servier Group company|Servier
 May 2025 Phase 1|Phase 2
NCT05992831 Recruiting
Mild Cognitive Impairment|Depression
Medical University of South Carolina|National Institute on Aging (NIA)
 July 15 2024 Not Applicable
NCT06223971 Recruiting
COVID Long-Haul
Johns Hopkins University|Radiological Society of North America
 May 20 2024 Early Phase 1
NCT06135064 Not yet recruiting
PTSD
University of Utah
 April 2024 Phase 1|Phase 2
NCT06223672 Recruiting
Cognitive Decline|Cognitive Impairment
Ohio State University|United States Department of Agriculture (USDA)|The California Walnut Commission
 February 7 2024 Not Applicable

Chemical Information & Solubility

Molecular Weight 333.46 Formula

C20H31NO3
CAS No. 77-23-6 SDF --
Density 1.048 g/mL
Smiles CCN(CC)CCOCCOC(=O)C1(CCCC1)C2=CC=CC=C2
Storage (From the date of receipt) 2 years -20°C liquid

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